Copper‐mediated Intermolecular C−H aminohalogenation of Indoles at Room Temperature
نویسندگان
چکیده
Abstract An efficient intermolecular C−H aminohalogenation of indoles with azoles and NXS (X = F, Cl, Br, I) has been developed. This mild protocol provides a straightforward entry to structurally valuable 2‐azolyl‐3‐halogenated in one single operation. In addition, this attractive route for the synthesis polyfunctionalized is great significance due product's versatile reactivity further transformations.
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ژورنال
عنوان ژورنال: Asian Journal of Organic Chemistry
سال: 2022
ISSN: ['2193-5815', '2193-5807']
DOI: https://doi.org/10.1002/ajoc.202200457